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Product Infomation
Product NameGSK3326595
CAS No.1616392-22-3
Molecular Weight

452.55

Formula

C₂₄H₃₂N₆O₃

SMILES

O=C(C)N1CCC(NC2=NC=NC(C(NC[C@H](O)CN3CCC(C=CC=C4)=C4C3)=O)=C2)CC1

Stock statusGet quote



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Product description

Description

GSK3326595 (EPZ015938) is a potent, selective, reversible inhibitor of protein arginine methyltransferase 5 (PRMT5) with an IC50 of 6.2 nM[1].



IC50 & Target

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IC50: 6.2 nM (PRMT5)[1]


In Vitro

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GSK3326595 (EPZ015938), has entered clinical trials for the treatment of solid tumors and non-Hodgkin’s lymphoma[1].





Powder-20°C3 years

4°C2 years
In solvent-80°C6 months

-20°C1 month







Peferences:

 [1]. WO 2016022605 A1